CAS NO:478082-99-4; ro4368554

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CAS:

478082-99-4

分子式:

C₁₉H₂₁N₃O₂S

分子量:

355.45

英文名称:

ro4368554

3-benzenesulfonyl-7-(4-methyl-piperazin-1-yl)-1h-indole

7-(4-methyl-1-piperazinyl)-3-(phenylsulfonyl)-1h-indole

用途:

Ro4368554 is a 5-HT6 receptor antagonist. RO4368554 acts selectively at 5-HT6 receptors where it binds with a greater than 100-fold selectivity over other monoamine receptor subtypes (-log M pKi = 9.4 at 5-HT6 and 7.1 at 5-HT2A).