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CAS: 1550053-02-5
分子式: C15H14FN3O2
分子量: 287.294
中文名称: 
4-乙酰胺基-n-(2-氨基-4-氟苯基)苯甲酰胺
英文名称: 
brd3308
4-acetamido-n-(2-amino-4-fluorophenyl)benzamide
用途: BRD3308 is a highly selective HDAC3 inhibitor with an IC50 of 54 nM. BRD3308 is 23-fold selectivity for HDAC3 over HDAC1 (IC50 of 1.26 μM) or HDAC2 (IC50 of 1.34 μM). BRD3308 suppresses pancreatic β-cell apoptosis induced by inflammatory cytokines or glucolipotoxic stress, and increases functional insulin release. BRD3308 activates HIV-1 transcription and disrupts HIV-1 latency[1][2][3].
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货号品牌产品名称规格包装、参考价格详情
B795726MACKLINBRD330810mM in DMSO466元/1ml;   展开
储存:-20°C
B910242MACKLINBRD330898%478元/50mg;   814元/100mg;   1381元/250mg;   4446元/1g;   展开
储存:-20°C,密闭,干燥
状态:白色固体
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