4-[2-(5-amino-1h-pyrazol-4-yl)-4-chloro-phenoxy]-5-chloro-2-fluoro-n-thiazol-4-yl-benzenesulfonamide p-toluene sulfonate salt
用途:
PF-05089771 is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 11 nM, >1,000-fold selectivity over Nav1.3, 1.4 and Nav1.5, 1.8.