CAS NO:1187020-80-9; 4-((6br,10as)-3-methyl-2,3,6b,9,10,10a-hexahydro-1h,7h-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-butan-1-one 4-methylbenzenesulfonate

CAS:

1187020-80-9

分子式:

C₃₁H₃₆FN₃O₄S

分子量:

565.7

中文名称:

4-((6br,10as)-3-methyl-2,3,6b,9,10,10a-hexahydro-1h,7h-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-butan-1-one 4-methylbenzenesulfonate

1-(4-fluorophenyl)-4-[(6br,10as)-3-methyl-2,3,6b,9,10,10a-hexahydro-1h-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7h)-yl]butan-1-one 4-methylbenzenesulfonate

英文名称:

lumateperone tosylate

iti-007

用途:

Lumateperone甲苯磺酸盐是5-HT 2A受体拮抗剂 (KI= 0.54 nM), 突触前D2受体的部分激动剂和突触后D2受体的拮抗剂 (KI= 32 nM)。